发明名称 Indolopyrrolocarbazole derivatives.
摘要 <p>Indolopyrrolocarbazole derivs. of formula (I) are new. In (I) R1, R2 = H, alkyl, alkenyl alkynyl, aryl, aralkyl or hetero (each opt. substd. by 1-5 of carboxy, carbamoyl, sulpho, NH2, CN, mono- and dialkylamino, OH and halo) or a gp. Y-R3; Y = carbonyl, thiocarbonyl of sulphonyl; R3 = H, alkyl, cycloalkyl, cycloalkylalkyl, aryl, aralkyl, hetero (each opt. substd. by 1-4 of halo, OH, carboxyl, CN, alkoxycarbonyl or NH2 and carbamoyl (each opt. substd. by 1-2 alkyl further substd. by halo, OH, NH2, carboxyl, carbamoyl and alkoxycarbonyl)) alkoxy, hydrazino, NH2, arylamino or carbamoyl; or R1 + R2 = alkidine opt. substd. by 1-4 of NH2, mono- or dialkylamino, OH, carboxyl and sulphonyl; or R1 + R2 = combined with the N to which they are attached form a heterocyclic gp. opt. substd. by alkyl further opt. substd. by NH2, Oh, carboxyl and sulpho; G = pentose or hexose; and X1, X2 = H, halo, NH2, mono- or dialkylamino, OH, alkoxy, aralkoxy carboxyl alkoxycarbonyl or alkyl.</p>
申请公布号 GR3018527(T3) 申请公布日期 1996.03.31
申请号 GR19950403667T 申请日期 1995.12.22
申请人 BANYU PHARMACEUTICAL CO., LTD. 发明人 KATSUHISA, KOJIRI;HISAO, KONDO;HIROHARU, ARAKAWA;OHKUBO, MITSURU;HIROYUKI, SUDA
分类号 C07D403/14;A61K31/40;A61K31/70;A61K31/7042;A61K31/7052;A61K31/7056;A61P35/00;C07D207/04;C07H19/044;C07H19/23;(IPC1-7):C07H19/044 主分类号 C07D403/14
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