发明名称 CONDENSED [1,4]DIAZEPINE COMPOUNDS AS AUTOTAXIN (ATX) AND LYSOPHOSPHATIDIC ACID (LPA) PRODUCTION INHIBITORS
摘要 wherein R1, R2, A1 and A2 are as described herein, compositions including the compounds and methods of using the compounds as autotaxin inhibitors.
申请公布号 SG11201607845R(A) 申请公布日期 2016.10.28
申请号 SG11201607845R 申请日期 2015.03.23
申请人 F. HOFFMANN-LA ROCHE AG 发明人 HUNZIKER, DANIEL;HERT, JÉRÔME;KUEHNE, HOLGER;MATTEI, PATRIZIO;RUDOLPH, MARKUS
分类号 C07D487/04;A61K31/551;A61P1/16;A61P3/00;A61P37/08 主分类号 C07D487/04
代理机构 代理人
主权项
地址