发明名称 |
CONDENSED [1,4]DIAZEPINE COMPOUNDS AS AUTOTAXIN (ATX) AND LYSOPHOSPHATIDIC ACID (LPA) PRODUCTION INHIBITORS |
摘要 |
wherein R1, R2, A1 and A2 are as described herein, compositions including the compounds and methods of using the compounds as autotaxin inhibitors. |
申请公布号 |
SG11201607845R(A) |
申请公布日期 |
2016.10.28 |
申请号 |
SG11201607845R |
申请日期 |
2015.03.23 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
HUNZIKER, DANIEL;HERT, JÉRÔME;KUEHNE, HOLGER;MATTEI, PATRIZIO;RUDOLPH, MARKUS |
分类号 |
C07D487/04;A61K31/551;A61P1/16;A61P3/00;A61P37/08 |
主分类号 |
C07D487/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|