发明名称 METHOD OF PREPARING ERGOALKALOIDS OF ERGOTOXINE AND ERGOTAMINE GROUP
摘要 FIELD: phytopreparations. SUBSTANCE: universal method of preparing ergot alkaloids is based on extraction with acid aqueous acetone solution, extract evaporation, conversion of ergoalkaloid salts to free bases by change of medium pH to alkaline value followed by extraction of total ergoalkaloids with chloroform, evaporation of chloroform extract to dry residue, dissolving obtained total ergoalkaloids in ethyl acetate, crystallization and filtration of ready product. Purity degree of ergoalkaloids is 96-98% at retained yield. EFFECT: simplified technology, enhanced purity.
申请公布号 RU94025607(A) 申请公布日期 1996.08.10
申请号 RU19940025607 申请日期 1994.07.07
申请人 NAUCHNO-PROIZVODSTVENNOE OB"EDINENIE "VSEROSSIJSKIJ NAUCHNO-ISSLEDOVATEL'SKIJ INSTITUT LEKARSTVENNYKH I AROMATICHESKIKH RASTENIJ";MEDITSINSKAJA AKADEMIJA IM.M.I.SECHENOVA 发明人 BYKOV V.A.;PETUKHOV S.A.
分类号 C07D457/02;C07D457/12 主分类号 C07D457/02
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