摘要 |
The invention relates to novel piperidine and pyrrolidine derivatives of formula (I) in which R<1>, R<2>, R<3>, k, l, m and n have the meanings indicated in Claim 1, and their salts, novel intermediates and processes for the preparation of the compounds according to the invention. The compounds of formula (I) act as 5-HT1A receptor antagonists and exhibit 5-HT reuptake-inhibiting actions and can be used for the production of medicaments. |
申请人 |
MERCK PATENT GMBH, 64293 DARMSTADT, DE |
发明人 |
ANDERSSON, BENGT RONNY, DIPL.-CHEM. DR., GOETEBORG, SE;HANSSON, LARS OLOV, DIPL.-CHEM. DR., GOETEBORG, SE;SONESSON, CLAS AKE, DIPL.-CHEM. DR., BILLDAL, SE;STJERNLOEF, NILS PETER, DIPL.-CHEM. DR., FROELIINDA, SE;MAERZ, JOACHIM, DIPL.-CHEM. DR., 55128 MAINZ, DE;BOETTCHER, HENNING, DIPL.-CHEM. DR., 64287 DARMSTADT, DE;DEVANT, RALF, DIPL.-CHEM. DR., 64291 DARMSTADT, DE;GREINER, HARTMUT, DIPL.-CHEM. DR., 64331 WEITERSTADT, DE;BARTOSZYK, GERD, DIPL.-PSYCH., 64331 WEITERSTADT, DE;HARTING, JUERGEN, DR., 64287 DARMSTADT, DE;SEYFRIED, CHRISTOPH, DIPL.-CHEM. DR., 64342 SEEHEIM-JUGENHEIM, DE |