发明名称 NOVEL IMINO DERIVATIVES AS INHIBITORS OF BONE RESORPTION ANDVITRONECTIN RECEPTOR ANTAGONISTS
摘要 Novel imino derivatives as inhibitors of bone resorption and vitronectin receptor antagonists There are described imino derivatives of the formula I R1-Y-A-B-D-E-F-G (I) in which R1, Y, A, B, D, E, F and G have the meaning indicated in the patent claims, their preparation and their use as medicaments. The compounds according to the invention are used as vitronectin receptor antagonists and as inhibitors of bone resorption.
申请公布号 CA2211148(A1) 申请公布日期 1998.01.24
申请号 CA19972211148 申请日期 1997.07.23
申请人 HOECHST AKTIENGESELLSCHAFT;GENENTECH, INC. 发明人 GOURVEST, JEAN-FRANCOIS;STILZ, HANS ULRICH;WEHNER, VOLKMAR;PITTI, ROBERT MAURICE;BODARY, SARAH CATHERINE;MCDOWELL, ROBERT;GADEK, THOMAS RICHARD;CARNIATO, DENIS;KNOLLE, JOCHEN
分类号 C07C229/04;A61K31/19;A61K31/197;A61K31/415;A61K31/445;A61P3/00;A61P9/00;A61P13/02;A61P15/00;A61P19/08;A61P27/02;A61P29/00;A61P35/00;A61P43/00;C07C251/02;C07D211/18;C07D233/52;C07D233/54;C07D233/66;C07D257/04;(IPC1-7):C07D233/52;C07D471/04;C07D249/14;C07D239/18;C07C279/22;A61K31/27;C07D235/30;A61K31/41;C07D239/42;A61K31/435;C07D277/50;A61K31/505;C07F9/547;A61K31/675;C07D213/77;C07D233/88 主分类号 C07C229/04
代理机构 代理人
主权项
地址