发明名称 POLYMORPHIC SALT OF AN ANTI-MIGRAIN DRUG.
摘要 THE PRESENT INVENTION IS CONCERNED WITH A CRYSTALLINE , POLYMORPHIC FORM OF A COMPOUND OF FORMULA (I) (FORMULA I)CHARACTERISED BY A POWDER X-RAY DIFFRACTION PATTERN OBTAINED USING COPPER K-ALPHA1 RADIATION (LAMBDA=0.15046NM) WHICH SHOWS MAIN PEAKS AT 9.28, 10.38, 11.37, 12.40, 16.84, 17.46, 17.53, 17.78, 19.48, 20.70, 21.45, 22.21, 22.64, 23.08, 25.20 AND 25.79.THE INVENTION ALSO RELATES TO PROCESSES FOR THE PREPARATION OF SAID FORM , TO PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND TO ITS USE IN MEDICINE , PARTICULARLY THE TREATMENT OF CONDITIONS FOR WHICH AN AGONIST OF 5-HT1 RECEPTORS IS INDICATED , FOR EXAMPLE , MIGRAINE.
申请公布号 MY121170(A) 申请公布日期 2005.12.30
申请号 MY2000PI04476 申请日期 2000.09.26
申请人 PFIZER INC. 发明人 ARTHUR BENTLEY;SIMON ARNOLD HOWARD-FIELD;RONALD JAMES OGILVIE
分类号 C07D403/06;A61K9/08;A61K9/20;A61K31/404;A61P1/08;A61P1/14;A61P3/04;A61P9/12;A61P25/06;A61P25/20;A61P25/24;A61P25/30;A61P29/00;A61P43/00 主分类号 C07D403/06
代理机构 代理人
主权项
地址