发明名称 TAXOIDS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 <p>TAXOIDS OF FORMULA: IN WHICH: Z REPRESENTS A HYDROGEN ATOM OR A RADICAL OF FORMULA: IN WHICH R1 REPRESENTS AN OPTIONALLY SUBSTITUTED BENZOYL RADICAL OR A THENOYL OR FUROYL RADICAL OR A RADICAL R2-O-CO- IN WHICH R2 REPRESENTS AN ALKYL, ALKENYL, ALKYNYL, CYCLOALKYL, CYCLOALKENYL, BICYCLOALKYL, OPTIONALLY SUBSTITUTED PHENYL OR HETEROCYCLIC RADICAL, R3 REPRESENTS AN ALKYL, ALKENYL, ALKYNYL, CYCLOALKYL, PHENYL, NAPHTHYL OR AROMATIC HETEROCYCLIC RADICAL, R4 REPRESENTS AN OPTIONALLY SUBSTITUTED ALKOXY, ALKENYLOXY OR ALKYNYLOXY RADICAL OR A CYCLOALKYLOXY OR CYCLOALKENYLOXY RADICAL, AND R5 REPRESENTS AN OPTIONALLY SUBSTITUTED ALKOXY, ALKENYLOXY OR ALKYNYLOXY RADICAL OR A CYCLOALKYLOXY OR CYCLOALKENYLOXY RADICAL ARE DESCRIBED: COMPOUNDS OF FORMULA (I) IN WHICH Z REPRESENTS A RADICAL OF FORMULA (II) DISPLAY NOTEWORTHY ANTITUMOUR AND ANTILEUKAEMIC PROPERTIES.</p>
申请公布号 MY121225(A) 申请公布日期 2006.01.28
申请号 MY1996PI01132 申请日期 1996.03.26
申请人 AVENTIS PHARMA S.A. 发明人 HERVE BOUCHARD;JEAN-DOMINIQUE BOURZAT;ALAIN COMMERCON
分类号 C07D305/14;A61K31/00;A61K31/335;A61K31/337;A61P35/00 主分类号 C07D305/14
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