发明名称 Halogen-substituted pyrazole derivatives as pest-control agents
摘要 The invention relates inter alia to halogen-substituted compounds of the general formula (I); in which the radicals A1-A4, T, n, W, Q, R1 and Z1-Z3 have the meanings given in the description. Also described are processes for preparing the compounds of the formula (I) and possible intermediates for the preparation of these compounds. The compounds according to the invention are particularly suitable for controlling insects, arachnids and nematodes in agriculture and ectoparasites in veterinary medicine.
申请公布号 US9487489(B2) 申请公布日期 2016.11.08
申请号 US201414762825 申请日期 2014.02.03
申请人 BAYER CROPSCIENCE AKTIENGESELLSCHAFT 发明人 Maue Michael;Ilg Kerstin;Decor Anne;Bretschneider Thomas;Hahn Julia Johanna;Hallenbach Werner;Fischer Reiner;Schwarz Hans-Georg;Goergens Ulrich;Raming Klaus;Koebberling Johannes;Huebsch Walter;Turberg Andreas;Lindner Niels
分类号 C07D401/12;C07D403/04;C07D231/12;C07D409/14;C07D401/14;C07D231/14;C07D403/14;C07D413/14;C07D231/18;A01N43/60;A01N43/713;A01N43/80;A01N43/82;A01N43/56 主分类号 C07D401/12
代理机构 McBee Moore Woodward Vanik IP LLC 代理人 McBee Moore Woodward Vanik IP LLC
主权项 1. Compound of formula (I), in which R1 represents hydrogen, optionally substituted C1-C6-alkyl, C3-C6-alkenyl, C3-C6-alkynyl, C3-C7-cycloalkyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, aryl-(C1-C3)-alkyl, or heteroaryl-(C1-C3)-alkyl, the chemical groupings A1 represents CR2 or nitrogen, A2 represents CR3 or nitrogen, A3 represents CR4 or nitrogen and A4 represents CR5 or nitrogen, but where not more than three of the chemical groupings A1 to A4 simultaneously represent nitrogen; R2, R3, R4 and R5 independently of one another represent hydrogen, halogen, cyano, nitro, optionally substituted C1-C6-alkyl, C3-C6-cycloalkyl, C1-C6-alkoxy, N—C1-C6-alkoxy-imino-C1-C3-alkyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl, N—C1-C6-alkylamino or N,N-di-C1-C6-alkylamino; if none of the groupings A2 and A3 represents nitrogen, R3 and R4 together with the carbon atom to which they are attached may form a 5- or 6-membered ring which contains 0, 1 or 2 nitrogen atoms and/or 0 or 1 oxygen atom and/or 0 or 1 sulphur atom, or if none of the groupings A1 and A2 represents nitrogen, R2 and R3 together with the carbon atom to which they are attached may form a 6-membered ring which contains 0, 1 or 2 nitrogen atoms; W represents oxygen or sulphur; Q represents hydrogen, formyl, hydroxy, amino or one of the optionally substituted groupings alkyl, alkyloxy, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, cycloalkylalkyl, arylalkyl, heteroarylalkyl or represents a grouping N-alkylamino, N-alkylcarbonylamino, N,N-dialkylamino; or Q represents an unsaturated 6-membered carbocycle which is optionally polysubstituted by V or an unsaturated 5- or 6-membered heterocyclic ring which is optionally polysubstituted by V, where V represents halogen, cyano, nitro, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, N-alkoxyiminoalkyl, alkylsulphanyl, alkylsulphinyl, alkylsulphonyl, or N,N-dialkylamino, T represents one of the 5-membered heteroaromatics T1-T7 listed below, where the bond to the pyrazole head group is marked with an asterisk, where R6 independently of one another represent halogen, cyano, nitro, amino or optionally substituted C1-C6-alkyl, C1-C6-alkyloxy, C1-C6-alkylcarbonyl, C1-C6-alkylsulphanyl, C1-C6-alkylsulphinyl, or C1-C6-alkylsulphonyl, and n represents the values 0-2; Z1 represents optionally substituted alkyl or cycloalkyl, and Z2 represents hydrogen, halogen, cyano, nitro, amino or optionally substituted alkyl, alkylcarbonyl, alkylsulphanyl, alkylsulphinyl, or alkylsulphonyl, and Z3 represents hydrogen or optionally substituted alkyl, cycloalkyl, alkenyl, alkynyl, aryl or hetaryl.
地址 Monheim DE
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