发明名称 |
N-acyl amino acid derivatives for treating skin conditions such as cellulite |
摘要 |
The invention relates to small molecules having biological and therapeutic activity. Particularly, the invention relates to small molecules having lipolytic and anti-adipogenic activity. Two examples of such molecules are 4-methyl-2-(octanoylamino) pentanoic acid and N-isopentyloctanamide. The invention further relates to methods of preventing or treating skin conditions such as cellulite using small molecules having lipolytic and anti-adipogenic activity. |
申请公布号 |
US9511042(B2) |
申请公布日期 |
2016.12.06 |
申请号 |
US201113703292 |
申请日期 |
2011.06.28 |
申请人 |
HELIX BIOMEDIX INC. |
发明人 |
Falla Timothy J.;Zhang Lijuan |
分类号 |
A61K8/44;A61K8/42;C07C237/12;A61K31/198;A61K31/20;A61Q19/06;A61K45/06 |
主分类号 |
A61K8/44 |
代理机构 |
Thomas Law PLLC |
代理人 |
Thomas Law PLLC |
主权项 |
1. A method of stimulating lipolysis in one or more adipocytes of a mammal, said method comprising administering to the skin tissue of said mammal a composition comprising a pharmaceutically acceptable carrier and a pharmaceutically effective amount of a compound, or salt thereof, wherein the compound is: |
地址 |
Bothell WA US |