发明名称 |
2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydoimidazo{1,2-a}pyrimidin-5(1H)one derivatives |
摘要 |
Imidazo[1,2-alpha]pyrimidinones and pyrimido[1,2-alpha]pyrimidinones useful for preventive and/or therapeutic treatment of neurodegenerative diseases, such as Alzheimer's disease, caused by abnormal GSK3beta activity. |
申请公布号 |
US6974819(B2) |
申请公布日期 |
2005.12.13 |
申请号 |
US20030362850 |
申请日期 |
2003.06.17 |
申请人 |
MITSUBISHI PHARMA CORPORATION |
发明人 |
GARCIA ANTONIO ALMARIO;GALLET THIERRY;LI ADRIEN TAK;LOCHEAD ALISTAIR;MARGUERIE SEVERINE;NEDELEC ALAIN;SAADY MOURAD;YAICHE PHILIPPE |
分类号 |
A61K31/519;A61P3/04;A61P3/10;A61P9/00;A61P9/10;A61P17/14;A61P23/02;A61P25/00;A61P25/02;A61P25/16;A61P25/24;A61P25/28;A61P27/06;A61P35/00;A61P35/02;C07D487/04;(IPC1-7):C07D487/04 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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