发明名称 Acetatic abiraterone trifluoroacetate and preparation method and application of same
摘要 Provided are acetaic abiraterone trifluoroacetate, a preparation method and an application of same. The acetaic abiraterone trifluoroacetate is obtained through a salt-forming reaction between acetaic Abiraterone and trifluoroacetic acid. The acetaic abiraterone trifluoroacetate undergoes self-purification through recrystallization, and dissociation and recrystallization are performed on the purified abiraterone acetate trifluoroacetate, so that the obtained acetaic abiraterone has a high purity, a high yield and stable quality, and is capable of meeting the requirement for mass production of acetaic abiraterone.
申请公布号 US9522934(B2) 申请公布日期 2016.12.20
申请号 US201314409791 申请日期 2013.02.20
申请人 Shanghai Cdymax Pharmaceuticals Co., Ltd.;Jiangsu Cdymax Pharmaceuticals Co., Ltd.;Shanghai Acebright Pharmaceuticals Group Co., Ltd. 发明人 An Xiaoxia;Huang Chengjun;Mao Fengwang
分类号 A61K31/4406;C07J43/00;C07C53/10 主分类号 A61K31/4406
代理机构 Hamre, Schumann, Mueller & Larson, P.C. 代理人 Hamre, Schumann, Mueller & Larson, P.C.
主权项 1. An abiraterone acetate trifluoroacetate, having the following chemical formula:
地址 Shanghai CN