发明名称 Synthesis of peptide aminoalkylamides and peptide hydrazides by the solid-phase method
摘要 The invention relates to compounds of the formula I <IMAGE> in which A denotes hydrogen or an amino protective group, B denotes one or more amino acids, X denotes alkylene or aralkylene, Y1, Y2, Y3 and Y4 are identical or different and denote hydrogen, methyl, methoxy or nitro, V denotes hydrogen or a carboxyl protective group, W denotes -[CH2]n- or -O-[CH2]n-, m denotes 0 or 1, n denotes 0 to 6, and p denotes 0 to 5, to a process for their preparation. The compounds of formula I are useful as linkage agents or anchor groups in the solid-phase synthesis of peptide aminoalkylamides and peptide hydrazides.
申请公布号 US5565606(A) 申请公布日期 1996.10.15
申请号 US19940257446 申请日期 1994.06.08
申请人 HOECHST AKTIENGESELLSCHAFT 发明人 BREIPHOL, GERHARD;KNOLLE, JOCHEN
分类号 A61K38/00;C07K1/04;C07K14/58;C07K14/60;(IPC1-7):C07C261/00 主分类号 A61K38/00
代理机构 代理人
主权项
地址