发明名称 HYDROXYETHYLAMINOSULFONAMIDE VERWENDBAR ALS INHIBITOREN RETROVIRALER PROTEASEN
摘要 The present invention provides retroviral protease inhibitor compounds represented by the Formula I: <CHEM> Such compounds are urseful for preparing medicaments for inhibiting proteases, especially for inhibiting HIV protease and for treating a retroviral infection such as HIV infection and for treating AIDS.
申请公布号 DE69321845(D1) 申请公布日期 1998.12.03
申请号 DE1993621845 申请日期 1993.08.24
申请人 G.D. SEARLE & CO., CHICAGO, ILL., US;MONSANTO CO. (N.D.GES.D.STAATES DELAWARE), ST. LOUIS, MO., US 发明人 VAZQUEZ, MICHAEL, L., GURNEE, IL 60031, US;MUELLER, RICHARD, A., GLENCOE, IL 60022, US;TALLEY, JOHN, J., CHESTERFIELD, MO 63017, US;GETMAN, DANIEL, CHESTERFIELD, MO 63017, US;DECRESCENZO, GARY, A., ST. PETERS, MO 63376, US;FRESKOS, JOHN, N., CLAYTON, MO 63105, US
分类号 C07D295/12;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4433;A61K31/505;A61K31/535;A61K31/5375;A61K38/00;A61P31/12;C07C311/05;C07C311/11;C07C311/13;C07C311/14;C07C311/18;C07C311/20;C07C311/24;C07C311/29;C07C311/32;C07C311/41;C07C311/46;C07C313/06;C07C317/04;C07C317/10;C07C317/14;C07C317/28;C07C317/44;C07C323/49;C07C323/57;C07C323/67;C07C327/38;C07D209/08;C07D211/78;C07D213/30;C07D213/53;C07D213/56;C07D213/64;C07D213/73;C07D213/81;C07D213/82;C07D213/89;C07D215/48;C07D233/54;C07D239/02;C07D239/26;C07D277/24;C07D277/30;C07D277/82;C07D307/20;C07D307/42;C07D307/79;C07D317/62;C07D333/34;C07D405/12;C07D409/12;C07D417/12;C07K5/06;C07K5/078;(IPC1-7):C07C311/29 主分类号 C07D295/12
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