发明名称 PROCESS FOR PREPARING HETEROCYDIC DERIVATIVES
摘要 A process for manufg. heterocyclic derivs. (I) used for effective antihistamines and antacids are described. Guanidine derivs (I; X = S or NH; Y = O or S; m = 0-4; n = 1-4; R1 = H, halo, C1-6 alkyl; R2 = H, C1-10 alkyl, C1-6 alkaloyl; A = 3,4-dioxocyclobutene-1,2 diol; B = C1-6 alkoxy) are prepd. by reacting compd. III and compd. IV.
申请公布号 KR810000600(B1) 申请公布日期 1981.06.05
申请号 KR19810001192 申请日期 1981.04.20
申请人 IMPERIAL CHEMICAL IND LTD;I C I AMERICAS INC 发明人 YELLIN T;WARDLEWORTH J;GILMAN D;JONES D
分类号 A61K31/415;A61K31/54;C07D233/88;C07D277/42;(IPC1-7):C07D277/42;A61K31/41 主分类号 A61K31/415
代理机构 代理人
主权项
地址