发明名称 1,3-DISUBSTITUTED OXIDOLES AND THE PROCESS
摘要 2-ox-indole compound, formula (I), or its salt is prepared by treating formula (IV) with acylisocyanate, R2-C(=O)-N=C=O, in inert solvent or formula (II) with activated derivative of carboxylic acid R1-C(=O)-OH, in inert solvent. In formula, X, Y represent a resonable C1-7 alkyl compound or a hetero compound, respectively, or halogen, hydrogen, or a combinded alkyl compound or a hetero compound, together. And R1, R2 are alkyl group having a resonable substituent, respectively.
申请公布号 KR880000433(B1) 申请公布日期 1988.03.24
申请号 KR19850000714 申请日期 1985.02.05
申请人 PFIZER INC. 发明人 KADIN, SAUL BERNARD
分类号 C07D495/04;A61K;A61K31/00;A61K31/33;A61K31/395;A61K31/40;A61K31/403;A61K31/404;A61K31/405;A61K33/00;A61P25/04;A61P29/00;A61P43/00;C07C;C07D;C07D209/00;C07D209/02;C07D209/32;C07D209/34;C07D209/38;C07D307/00;C07D333/00;C07D405/06;C07D405/12;C07D407/06;C07D409/06;C07D409/12;C07D491/048;C07D491/056;(IPC1-7):C07D209/32 主分类号 C07D495/04
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