发明名称 COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
摘要 The present invention relates to compounds of formula I. The compounds are inhibitors of the Src Homolgy-2 phosphatase (SHP2) and thus useful in the treatment of Noonan Syndrome, Leopard Syndrome and cancer.
申请公布号 WO2016203406(A1) 申请公布日期 2016.12.22
申请号 WO2016IB53550 申请日期 2016.06.15
申请人 NOVARTIS AG;CHEN, Zhuoliang;FORTANET, Jorge Farcia;JOUK, Andriana;KARKI, Rajesh;LAMARCHE, Matthew J.;LIU, Gang;PALERMO, Mark G.;PEREZ, Lawrence Blas;SARVER, Patrick James;SHULTZ, Michael David;SENDZIK, Martin;TOURE, Bakary-Barry;YU, Bing 发明人 CHEN, Zhuoliang;FORTANET, Jorge Farcia;JOUK, Andriana;KARKI, Rajesh;LAMARCHE, Matthew J.;LIU, Gang;PALERMO, Mark G.;PEREZ, Lawrence Blas;SARVER, Patrick James;SHULTZ, Michael David;TOURE, Bakary-Barry;YU, Bing
分类号 C07D401/14;A61K31/506;A61K31/537;A61P9/00;A61P19/00;A61P21/00;A61P25/28;A61P35/00;C07D401/04;C07D471/10;C07D491/107;C07D498/10 主分类号 C07D401/14
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