| 主权项 |
1. A compound of formula (I) wherein B is C1-C4-alkylene, C2-C4-alkenylene, C2-C4-alkynylene, —O—(C1-C4-alkylene)-,—S—(C1-C4-alkylene)-;
R is selected from the group consisting of: R1 and R2 together with the nitrogen atom to which they are attached, form a bicyclic ring system or heterocycloalkyl which can be substituted by 1 to 3 substituents independently selected from the group consisting of halogen, C1-C7-alkyl, C1-C7-hydroxyalkyl, C1-C7 alkoxy, C1-C7-haloalkyl, hydroxyl and oxo; R3 is selected from hydrogen, C1-C7-alkyl, C1-C7-alkoxyalkyl, C1-C7-haloalkyl, (CH2)1,2—C3-C5-cycloalkyl, —(CH2)1,2-aryl optionally substituted by C1-C7 alkoxy; R4 and R5 are independently selected from hydrogen, halogen, C1-C7-alkyl, C1-C7-haloalkyl, C1-C7-hydroxyalkyl, cyano, or R4 and R5 together form a C3-C8 cycloalkyl R6 is selected from hydrogen, C1-C7-alkyl, C1-C7-haloalkoxy, C3-C8 cycloalkyl, C1-C7 alkoxy, hydroxyl, halogen, S(O)2—C1-C7-alkyl, —C(O)NR′R″, NR′R″ wherein R′ and R″ are independently selected from hydrogen, C1-C7-alkyl or R′ and R″ together with the nitrogen atom to which they are attached from a heterocycloalkyl or R6 and R7 together form a C3-C8cycloalkyl, X is C—R7 wherein R7 is selected from hydrogen, C1-C7-alkyl, C1-C7 alkoxy, C1-C7-haloalkyl, C3-C8 cycloalkyl, —C(O)NR′R″ wherein R′ and R″ are independently selected from hydrogen and C1-C7-alkyl, Y is N or C—R4. |
