发明名称 Platform drug delivery system utilizing crystal engineering and theanine dissolution
摘要 A platform drug delivery system and a method of improving the delivery of low solubility pharmaceuticals utilizing crystal engineering and Theanine dissolution resulting in enhanced bioactivity, dissolution rate, and solid state stability.
申请公布号 US9603937(B2) 申请公布日期 2017.03.28
申请号 US201514642191 申请日期 2015.03.09
申请人 Theaprin Pharmaceuticals Inc. 发明人 Brittain Harry G.;Felice Philip V.
分类号 A61K47/18;A61K47/48;A61K31/704;A61K31/13;A61K31/137;A61K31/192;A61K31/198;A61K31/277;A61K31/4045;A61K31/4164;A61K31/4196;A61K31/426;A61K31/43;A61K31/445;A61K31/4745;A61K31/48;A61K31/496;A61K31/4985;A61K31/506;A61K31/522;A61K31/536;A61K31/545;A61K31/546;A61K31/549;A61K31/573;A61K31/635;A61K31/7048;A61K31/7072;A61K38/12 主分类号 A61K47/18
代理机构 Nataro, Michalos & Zaccaria P.C. 代理人 Nataro, Michalos & Zaccaria P.C.
主权项 1. A cocrystal of L-theanine; and doxorubicin, wherein said cocrystal is characterized as having an X-ray powder diffraction pattern with peaks (2θ) at 13.6, 18.2, 19.8, 22.0, 22.5, 25, and 38.2 degrees.
地址 Hauppauge NY US