| 摘要 |
The present invention provides the following compound having anti-HIV activity of formula:
wherein, A 1 is C, CR 1A or N;
A 2 is C, CR 2A , or N;
A 3 is CR 3A , CR 3A R 3B , N, NR 3c O, S, SO, or SO 2 ;
A 4 is CR 4A , CR 4A R 4B , N, NR 4C O, S, SO, or SO2;
A 5 is C, CR 5A , or N;
T 1 ring is substituted or unsubstituted monocyclic carbocycle or substituted or unsubstituted monocyclic heterocycle;
R 1 is halogen, cyano, nitro or -X 1 -R 11 ;
R 2 is substituted or unsubstituted alkyl and the like;
n is 1 or 2;
R 3 is hydrogen, substituted or unsubstituted aromatic varbocyclyl;
R 4 is hydrogen or a carboxy protecting group;
the other symbols are as specified in the description. |
