发明名称 PROCESS FOR RILPIVIRINE
摘要 The present invention provides a novel process for the preparation of 4-(4-hydroxypyrimidin-2-ylamino)benzonitrile. The present invention also provides a novel process for the preparation of 4-iodo-2,6-dimethyl benzenamine. The present invention further provides an improved process for the preparation of rilpivirine. The present invention further provides a tosylate salt of rilpivirine, process for its preparation and pharmaceutical compositions comprising it.
申请公布号 EP2702044(B1) 申请公布日期 2017.03.22
申请号 EP20120777741 申请日期 2012.02.16
申请人 Hetero Research Foundation 发明人 PARTHASARADHI REDDY, Bandi;RATHNAKAR REDDY, Kura;MURALIDHARA REDDY, Dasari;VENKAT NARSIMHA REDDY, Adulla;VAMSI KRISHNA, Bandi
分类号 C07D239/42 主分类号 C07D239/42
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