发明名称 PROCESS FOR THE PREPARATION OF SELEXIPAG AND INTERMEDIATES THEREOF
摘要 The present invention provides processes for the preparation of Selexipag compound of formula (1). The present invention also provides processes for the preparation of 4-[(5,6-diphenyl-pyrazin-2-yl)-isopropyl -amino]-butan-1-ol (2), and 4-isopropylamino-butan-1-ol of formula (3), which are intermediates for the synthesis of Selexipag (1 ).
申请公布号 WO2017042828(A2) 申请公布日期 2017.03.16
申请号 WO2016IN00226 申请日期 2016.09.07
申请人 MEGAFINE PHARMA (P) LTD. 发明人 MATHAD VIJAYAVITTHAL THIPPANNACHAR;DODDAPPA PRALHAD ANEKAL;KARDILE PRITESH BHIMRAJ;PADAKI SANTHOSH AMBADAS;GAIKWAD BAPUSAHEB SHRIHARI;SHINDE GORAKSHANATH BALASAHEB
分类号 C07D241/20;C07D239/42;C07D241/12;C07D241/18 主分类号 C07D241/20
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