发明名称 METHOD FOR PRODUCTING THIOLANE SKELETON-TYPE GLYCOCONJUGATE, AND THIOLANE SKELETON-TYPE GLYCOCONJUGATE
摘要 There is provided a production method of a compound represented by the following formula (II) through a step of reacting a compound represented by the following General Formula (I) with a sulfur compound. In General Formulas (I) and (II), R 1 represents a hydrogen atom or an acyl group, R 2 represents a hydrogen atom, a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R 3 represents a hydrogen atom or an acyloxy group, R 5 represents an alkyl group or an aryl group, and X represents a leaving group. Here, in a case where R 2 is a fluorine atom, an acyloxy group, an arylmethyloxy group, an allyloxy group, an arylmethyloxycarbonyloxy group, or an allyloxycarbonyloxy group, R 3 is an acyloxy group.
申请公布号 EP3109245(A4) 申请公布日期 2017.03.01
申请号 EP20150751503 申请日期 2015.02.17
申请人 FUJIFILM Corporation 发明人 ITO, Takayuki;WATANABE, Toru;OKADA, Hideki;KUNIYOSHI, Hidenobu
分类号 C07H1/00;C07D333/32;C07H13/08;C07H15/04;C07H15/18 主分类号 C07H1/00
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