发明名称 |
METHOD FOR THE PREPARATION OF (4S)-4-(4-CYANO-2-METHOXYPHENYL)-5-ETHOXY-2,8-DIMETHYL-1,4-DIHYDRO-1-6-NAPHTHYRIDINE-3-CARBOX-AMIDE AND THE PURIFICATION THEREOF FOR USE AS AN ACTIVE PHARMACEUTICAL INGREDIENT |
摘要 |
The invention relates to a new and improved method for preparing (4S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carbox-amide of formula (I) and to the production and use of the crystalline modification I of (4S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carbox-amide of formula (I). |
申请公布号 |
SG11201700785U(A) |
申请公布日期 |
2017.02.27 |
申请号 |
SG11201700785U |
申请日期 |
2015.07.29 |
申请人 |
BAYER PHARMA AKTIENGESELLSCHAFT |
发明人 |
PLATZEK, JOHANNES;GARKE, GUNNAR;GRUNENBERG, ALFONS |
分类号 |
C07D471/04;A61K31/4375;A61P9/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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