发明名称 HETEROARYL PIPERIDINE AND HETEROARYL PIPERAZINE DERIVATIVES AS FUNGICIDES
摘要 Heteroarylpiperidine and -piperazine derivatives of the formula (I);;in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).
申请公布号 US2017044153(A1) 申请公布日期 2017.02.16
申请号 US201615339576 申请日期 2016.10.31
申请人 BAYER INTELLECTUAL PROPERTY GMBH 发明人 HILLEBRAND Stefan;CRISTAU Pierre;HOFFMANN Sebastian;KLUTH Joachim;WASNAIRE Pierre;TSUCHIYA Tomoki;BENTING Juergen;WACHENDORFF-NEUMANN Ulrike;SEITZ Thomas
分类号 C07D417/14;A01N43/80 主分类号 C07D417/14
代理机构 代理人
主权项 1. A compound of the formula (I)in which the radicals are each defined as follows: A is phenyl which may contain up to two substituents, where the substituents are each independently selected from the following list: halogen, cyano, hydroxyl, —NR3R4, —C(═O)NR3R4, nitro, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C1-C6-haloalkyl, C2-C6-haloalkenyl, C2-C6-haloalkynyl, C3-C6-halocycloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkenyloxy, C1-C4-alkynyloxy, C1-C4-alkylthio, C1-C4-alkylsulphonyl, C1-C4-haloalkylthio, C1-C4-haloalkylsulphonyl, C1-C4-alkoxy-C1-C6-alkyl, hydroxy-C1-C4-alkyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, C1-C6-alkylcarbonyloxy or —C(═O)H, or A is a heteroaromatic radical selected from the following group: furan-2-yl, furan-3-yl, thiophen-2-yl, thiophen-3-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, pyrrol-1-yl, pyrrol-2-yl, pyrrol-3-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, pyrazol-1-yl, pyrazol-3-yl, pyrazol-4-yl, imidazol-1-yl, imidazol-2-yl, imidazol-4-yl, 1,2,3-triazol-1-yl, 1,2,4-triazol-1-yl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyridazin-3-yl, pyridazin-4-yl, pyrazin-2-yl, pyrazin-3-yl, pyrimidin-2-yl, pyrimidin-4-yl or pyrimidin-5-yl which may contain up to two substituents, where the substituents are each independently selected from the following list: substituents on carbon:halogen, cyano, hydroxyl, nitro, —NR3R4, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, C1-C6-haloalkyl, C2-C6-haloalkenyl, C2-C6-haloalkynyl, C3-C6-halocycloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-alkylsulphonyl, C1-C4-haloalkylthio, C1-C4-haloalkylsulphonyl, C1-C4-alkoxy-C1-C4-alkyl, hydro xy-C1-C4-alkyl, C1-C6-alkylcarbonyl, C1-C6-alkoxycarbonyl, C1-C6-alkylcarbonyloxy or phenyl, substituents on nitrogen: C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C6-haloalkyl, C2-C6-haloalkenyl, C2-C6-haloalkynyl, C3-C10-cycloalkyl-C1-C6-alkyl, C1-C6-haloalkylcarbonyl, phenyl, benzyl, C1-C4-alkylsulphonyl, C1-C4-haloalkylsulphonyl, phenylsulphonyl, —C(═O)H, or C1-C6-alkylcarbonyl, L1 is —NH—, Y is oxygen, X is carbon, R2 is hydrogen, p is 0, G is where the bond identified by “v” is bonded directly to X and where the bond identified by “w” is bonded directly to Q, RG1 is hydrogen, Q is R5 is hydrogen, L2 is a direct bond, where the bond identified by “x” is bonded directly to G, and the bond identified by “y” is bonded directly to L2, R1 is phenyl which is substituted once by a Z4 substituent and may additionally optionally have further substitution, where the additional substituents are each independently selected from Z4 and Z1-1, Z4 is C(═O)H, C1-C3-alkoxy-C2-C3-alkoxy-C1-C3-alkyl, C1-C4-alkylsulphinyl-C1-C2-alkyl, C1-C4-alkylsulphonyl-C1-C2-alkyl, C1-C4-haloalkoxy-C1-C2-alkyl, C3-C6-cycloalkyl-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C4-alkoxy-C1-C4-alkoxy, C3-C6-cycloalkylcarbonyloxy or C1-C4-alkylsulphonylamino, Z1-1 is halogen, C1-C6-alkyl, or C1-C6-haloalkyl; and/or a salt, metal complex and/or and N-oxide thereof.
地址 Monheim am Rhein DE