| 发明名称 |
FATTY ACID CONJUGATES OF QUETIAPINE, PROCESS FOR MAKING AND USING THE SAME |
| 摘要 |
The presently described technology provides a novel class of prodrugs of quetiapine that can be synthesized by chemically conjugating fatty acids to quetiapine. Pharmaceutical compositions and methods of synthesizing conjugates of the present technology are also provided. Methods of treating patients with the compositions of the present technology are also provided. |
| 申请公布号 |
US2017042906(A1) |
申请公布日期 |
2017.02.16 |
| 申请号 |
US201615340533 |
申请日期 |
2016.11.01 |
| 申请人 |
KemPharm, Inc. |
发明人 |
Mickle Travis;Guenther Sven;Bera Sanjib |
| 分类号 |
A61K31/554;A61K9/00;A61K45/06;A61K47/48 |
主分类号 |
A61K31/554 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
1. A composition for treating a psychiatric disorder in a subject, comprising:
2-(2-(4-(dibenzo[b,f][1,4]thiazepin-11-yl)piperazin-1-yl)ethoxy)ethanol (quetiapine) conjugated to capric acid, a salt of the conjugate or their combination. |
| 地址 |
Celebration FL US |
