Prodrugs of glutamine analogs, such as prodrugs of aza-serine, and 6-diazo-5-oxo-norleucine (DON), and 5-diazo-4-oxo-L-norvaline (L-DONV) are disclosed.
申请公布号
WO2017023774(A1)
申请公布日期
2017.02.09
申请号
WO2016US44767
申请日期
2016.07.29
申请人
THE JOHNS HOPKINS UNIVERSITY;INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY AS CR V.V.I.
发明人
SLUSHER, Barbara;RAIS, Rana;TENORA, Lukas;MAJER, Pavel;JANCARIK, Andrej;NEDELCOVYCH, Mike