Disclosed are mild temperature (e.g., from 0 to 80°C) SNAr fluorinations of a variety of halide and sulfonate substituted aryl and heteroaryl substrates using NMe4F.
申请公布号
WO2017024167(A1)
申请公布日期
2017.02.09
申请号
WO2016US45624
申请日期
2016.08.04
申请人
DOW AGROSCIENCES LLC;THE REGENTS OF THE UNIVERSITY OF MICHIGAN
发明人
SANFORD, Melanie;RYAN, Sarah;SCHIMLER, Sydonie;CHENG, Yang;BLAND, Douglas