发明名称 |
Fremgangsmåde til fremstilling af voriconazol og analoger deraf |
摘要 |
The present invention provides a process for preparing a compound of formula: (Formula XI and XII) (XI) (XII) wherein X, Y, Z, A, B and E are as defined herein, by reacting a compound of formula: (Formula XIII) (XIII) with a compound of formula: (Formula XIV and XV) (XIV) (XV) respectively, in the presence of a transition metal catalyst, a ligand suitable for use with 15 the catalyst and a reducing agent. The invention also provides novel intermediates. |
申请公布号 |
DK2906555(T3) |
申请公布日期 |
2017.02.06 |
申请号 |
DK20130795583T |
申请日期 |
2013.10.08 |
申请人 |
Pfizer Ireland Pharmaceuticals |
发明人 |
PETTMAN, Alan, John;BURRELL, Adam, James, Musgrave;O'NEILL, Padraig, Mary |
分类号 |
C07D403/06;C07D239/30 |
主分类号 |
C07D403/06 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|