发明名称 ONE POT PROCESS FOR PRODUCING 6-HYDROXYL NAL-OPIATE
摘要 The present invention provides processes for preparing nal-opiates without the isolation of intermediates. In general, the process provides for alkylation and reduction in the same pot to give the nal-opiate.
申请公布号 EP2812336(B1) 申请公布日期 2017.02.01
申请号 EP20130706352 申请日期 2013.02.08
申请人 Mallinckrodt LLC 发明人 WANG, Peter, X.;JIANG, Tao;BERBERICH, David, W.
分类号 C07D489/02;A61K31/485;C07D489/08 主分类号 C07D489/02
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