| 发明名称 |
METHOD FOR PRODUCING 4-BORONO-L-PHENYLALANINE HAVING 18F ATOM INTRODUCED THEREINTO, AND PRECURSOR OF 4-BORONO-L-PHENYLALANINE HAVING 18F ATOM INTRODUCED THEREINTO |
| 摘要 |
18F-labeled 4-boronophenylalanine (BPA) can be produced by preparing and further processing a precursor of 18F-labeled BPA represented by the following formula:;in which R1 represents a bromo group, an iodo group, a fluoro group, a diazaborinane derivative, BX3− or BX3−M+ (wherein X represents a halogen atom; and M+ represents a monovalent monoatomic cation, a polyatomic cation or a complex cation). |
| 申请公布号 |
US2017015684(A1) |
申请公布日期 |
2017.01.19 |
| 申请号 |
US201515122118 |
申请日期 |
2015.01.28 |
| 申请人 |
STELLA PHARMA CORPORATION ;OSAKA PREFECTURE UNIVERSITY PUBLIC CORPORATION |
发明人 |
TAKENAKA Hiroshi;OHTA Yoichiro;TAGUCHI Yusuke;UEDA Sayuri;ISHINO Yuko;YOSHIKAWA Tomohiro;NAKASHIMA Hideki;UEHARA Kohki;KIRIHATA Mitsunori |
| 分类号 |
C07F5/02;C07B59/00;C07C47/55;C07C45/63 |
主分类号 |
C07F5/02 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
1. A compound represented by a formula below: wherein R1 represents bromo group, iodo group, fluoro group, a diazaborinane derivative, BX3−, or BX3−M+ (X represents halogen, and M+ represents monovalent monoatomic cation, polyatomic cation, or complex cation). |
| 地址 |
Osaka JP |
