发明名称 PROCESS FOR PRODUCING HETEROCYCLIC COMPOUND
摘要 The present invention provides a method of efficiently producing an optically active 6-(3-aminopiperidin-1-yl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine derivative. The optically active piperidine-3-carboxamide or a derivative thereof, which is obtained by subjecting 1,4,5,6-tetrahydropyridine-3-carboxamide or a derivative thereof to an asymmetric reduction in the presence of a catalyst, is used as an intermediate.
申请公布号 EP3118192(A1) 申请公布日期 2017.01.18
申请号 EP20150762433 申请日期 2015.03.13
申请人 Takeda Pharmaceutical Company Limited 发明人 YAMADA, Masatoshi;HIRANO, Sayuri;TSURUOKA, Ryoji;YAMANO, Mitsuhisa
分类号 C07D211/60;B01J23/46;B01J23/70;C07B53/00;C07B61/00;C07D211/72;C07D401/04;C07F9/50;C07F15/00;C07F15/02 主分类号 C07D211/60
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