发明名称 THIAZOLE-SUBSTITUTED AMINOHETEROARYLS AS SPLEEN TYROSINE KINASE INHIBITORS
摘要 The invention provides certain thiazole-substituted aminoheteroaryl compounds of the Formula (I) (I), or pharmaceutically acceptable salts thereof, wherein ring R1, R2, R3, R4, ring A, and the subscripts n1, n2, and r are as defined herein. The invention also provides pharmaceutical compositions comprising such compounds, and methods of using the compounds for treating diseases or conditions mediated by Spleen Tyrosine Kinase (Syk).
申请公布号 EP3083560(A1) 申请公布日期 2016.10.26
申请号 EP20140872688 申请日期 2014.12.18
申请人 MERCK SHARP & DOHME CORP. 发明人 MILLER, THOMAS A.;PETROCCHI, ALESSIA;ROMEO, ERIC T.;VITHARANA, DILRUKSHI;KATTAR, SOLOMON D.;NORTHRUP, ALAN B.;ALTMAN, MICHAEL D.;ANTHONY, NEVILLE J.
分类号 C07D213/72 主分类号 C07D213/72
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