发明名称 CRYSTALLINE FORM OF (S)-(2-(6-CHLORO-7-METHYL-1H-BENZO[D]IMIDAZOL-2-YL)-2-METHYLPYRROLIDIN-1 -YL)(5-METHOXY-2-(2H-1,2,3-TRIAZOL-2-YL)PHENYL)METHANONE AND ITS USE AS OREXIN RECEPTOR ANTAGONISTS
摘要 The invention relates to crystalline forms of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone, processes for the preparation thereof, pharmaceutical compositions containing such crystalline forms, pharmaceutical compositions prepared from such crystalline forms, and their use as a medicament, especially as orexin receptor antagonists.
申请公布号 EP3077389(A1) 申请公布日期 2016.10.12
申请号 EP20140824107 申请日期 2014.12.02
申请人 ACTELION PHARMACEUTICALS LTD. 发明人 BOSS, CHRISTOPH;BROTSCHI, CHRISTINE;GUDE, MARKUS;HEIDMANN, BIBIA;SIFFERLEN, THIERRY;VON RAUMER, MARKUS;WILLIAMS, JODI, T.
分类号 C07D403/14;A61K31/4192;A61P25/00 主分类号 C07D403/14
代理机构 代理人
主权项
地址