发明名称 IMIDAZO[1,5]NAPHTHYRIDINE COMPOUNDS, THEIR PHARMACEUTICAL USE AND COMPOSITIONS
摘要 The present invention is directed to compounds of Formula (I), and to salts thereof, their synthesis, and their use as PI3-Kα inhibitors and/or PI3-Kα/mTOR dual inhibitors.
申请公布号 EP2356120(B1) 申请公布日期 2016.10.12
申请号 EP20090787247 申请日期 2009.09.18
申请人 PFIZER INC. 发明人 CHENG, HENGMIAO;JOHNSON, TED WILLIAM;HOFFMAN, JACQUI ELIZABETH;GUO, LISA CHEN;LIU, ZHENGYU;JOHNSON, THEODORE OTTO;LIU, KEVIN KUN-CHIN
分类号 C07D471/14;A61K31/33;A61P35/00 主分类号 C07D471/14
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