发明名称 AMORPHOUS ALLISARTAN ISOPROXIL, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION CONTAINING AMORPHOUS ALLISARTAN ISOPROXIL
摘要 The present invention relates to an amorphous allisartan isoproxil which is an angiotensin II receptor blocker with good flowability and a large bulk density and with no obvious electrostatic phenomenon; the find of the amorphous allisartan isoproxil can effectively reduce the generation of dust pollution during the production, thereby providing convenience the production of allisartan isoproxil. The present invention also relates to a pharmaceutical composition containing the amorphous allisartan isoproxil. The pharmaceutical composition is highly stable, and allisartan isoproxil formulation prepared from the pharmaceutical composition can effectively ensure the quality of the drug.
申请公布号 EP3064496(A1) 申请公布日期 2016.09.07
申请号 EP20140856893 申请日期 2014.10.29
申请人 SHENZHEN SALUBRIS PHARMACEUTICALS CO., LTD. 发明人 TAN,DUANMING;OU, JUN;YE, GUANHAO;BU, SHUI
分类号 C07D403/10;A61K31/4178;A61P9/12 主分类号 C07D403/10
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