发明名称 |
N-CYCLOPROPYL-N-PIPERIDINYLBENZAMIDES AS GPR119 MODULATORS |
摘要 |
The present invention relates to compounds of general formula I, wherein the groups R1, LP, LQ, Ar, m and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity. |
申请公布号 |
EP2686312(B1) |
申请公布日期 |
2016.08.31 |
申请号 |
EP20120708044 |
申请日期 |
2012.03.13 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
HECKEL, ARMIN;BLUM, ANDREAS;BREITFELDER, STEFFEN;HIMMELSBACH, FRANK;LANGKOPF, ELKE;NOSSE, BERND;WELLENZOHN, BERND;ASHWEEK, NEIL, J.;HARRIOTT, NICOLE |
分类号 |
C07D401/14;A61K31/41;A61K31/422;A61K31/4245;A61K31/454;A61P3/10;C07D413/14;C07D417/14 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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