发明名称 SOLID FORM OF PYRAZOLOPYRIDINE COMPOUND
摘要 A novel crystalline form or amorphous of formula (I) and preparation method thereof are disclosed in present invention, wherein the novel crystalline form is substantially pure crystalline form I, form II, form III or form IV. The novel crystalline forms disclosed herein have good solubility, low hydroscopicity and good stability at high temperature (60° C.), high humidity (RH is 90%±5%) and/or under light (4500+/−500 Lux), which benefit for storage, meet the requirements of drug stability and therefore, making formula (I) suitable for formulation preparation and with high bioavailability.
申请公布号 EP3057968(A1) 申请公布日期 2016.08.24
申请号 EP20140853930 申请日期 2014.10.15
申请人 SUNSHINE LAKE PHARMA CO., LTD. 发明人 LIAO, SHOUZHU;FAN, WEIJIE;WANG, ZHONGQING
分类号 C07D471/04;A61K31/506;A61P7/02;A61P9/00;A61P9/10;A61P9/12;A61P15/00 主分类号 C07D471/04
代理机构 代理人
主权项
地址