发明名称 INTERMEDIATES IN THE PREPARATION OF A BIS(BENZIMIDAZOLE)CYCLOPHANE DERIVATIVE
摘要 Provided is a compound having a structure selected from the group consisting of: which are intermediates in the preparation of Carbamic acid, N,N'-[tricyclo[8.2.2.24,7]hexadeca-4,6,10,12,13,15-hexaene-5,11-diyl bis [1H-benzimidazole-6,2-diyl[(2S,3aS,7aS)-octahydro-1H-indole-2,1-diyl][(1S)-1-(1-methylethyl)-2-oxo-2,1-ethane diyl]]] bis-, C,C'-dimethyl ester, which is a Hepatitis C virus NS5a (HCV NS5a) protease replication inhibitor
申请公布号 EP3059241(A1) 申请公布日期 2016.08.24
申请号 EP20160157270 申请日期 2012.05.29
申请人 ACHILLION PHARMACEUTICALS, INC. 发明人 WILES, JASON ALLAN;WANG, QIUPING;HASHIMOTO, AKIHIRO;PAIS, GODWIN;CHEN, DAWEI;WANG, XIANGZHU;GADHACHANDA, VENKAT;PHADKE, AVINASH;DESHPANDE, MILIND
分类号 C07F17/02;A61K31/4164;A61K31/4178;A61P31/00;A61P31/12;C07D401/14;C07D403/14;C07D413/14;C07D417/14;C07D471/08;C07D471/14;C07D491/10;C07D519/00 主分类号 C07F17/02
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