发明名称 |
NOVEL PYRAZOLE DERIVATIVE |
摘要 |
It has been desired to develop a pharmaceutical composition, which is used in agents for preventing and/or treating various diseases related to PDE10 (e.g. mental disorder and neurodegenerative disorder). The present invention provides: compounds having PDE10 inhibitory effect, in particular, compounds having a 4-heteroarylpyrazole-5-carboxylic acid amide structure represented by the following formula (I), or their pharmaceutically acceptable salts, or their solvates; pharmaceutical compositions comprising, as active ingredients, the compounds, or their pharmaceutically acceptable salts, or their solvates; and medical use of the compounds, or their pharmaceutically acceptable salts, or their solvates. |
申请公布号 |
EP2963037(A4) |
申请公布日期 |
2016.08.03 |
申请号 |
EP20140756804 |
申请日期 |
2014.02.26 |
申请人 |
MOCHIDA PHARMACEUTICAL CO., LTD. |
发明人 |
OKANO, AKIHIRO;SAITOH, FUMIHIKO;MAKABE, MUNEYOSHI;OGAWA, KOUKI |
分类号 |
C07D471/04;A61K31/444;A61K31/497;A61K31/506;A61K31/5377;A61P3/04;A61P25/00;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/32;A61P25/36;A61P43/00;C07D401/04;C07D403/04;C07D417/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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