发明名称 PROCESS FOR THE PURIFICATION OF DAPAGLIFLOZIN
摘要 The present invention provides a process for the preparation of (1C)-2,3,4,6-tetra-O-acetyl-1,5-anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-D-glucitol of Formula III. The invention also provides a process for the purification of dapagliflozin using (1C)-2,3,4,6-tetra-O-acetyl-1,5-anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-D-glucitol of Formula III.
申请公布号 EP3049397(A1) 申请公布日期 2016.08.03
申请号 EP20140784525 申请日期 2014.09.19
申请人 SUN PHARMACEUTICAL INDUSTRIES LTD 发明人 JAYACHANDRA, SURESH, BABU;NAGDA, DEVENDRA, PRAKASH;SINGH, TARUN, KUMAR
分类号 C07D309/10;C07H7/04 主分类号 C07D309/10
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