发明名称 |
METHOD FOR PRODUCING PYRROLE DERIVATIVE, AND INTERMEDIATE THEREOF |
摘要 |
The present invention provides a method for producing an atropisomer of a pyrrole derivative having excellent mineralocorticoid receptor antagonistic activity, and an intermediate thereof. A method for producing an atropisomer of a pyrrole derivative using a compound represented by (B) [wherein R 1 represents a C1-C4 alkyl group, and R 2 represents a 2-hydroxyethyl group or a carboxymethyl group] as a production intermediate. |
申请公布号 |
EP3040330(A1) |
申请公布日期 |
2016.07.06 |
申请号 |
EP20140839943 |
申请日期 |
2014.08.26 |
申请人 |
DAIICHI SANKYO COMPANY, LIMITED |
发明人 |
WATANABE, MASASHI;NAGASAWA, HIROSHI;SATO, NORITADA |
分类号 |
C07D207/456;C07B57/00;C12P41/00 |
主分类号 |
C07D207/456 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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