发明名称 METHOD FOR PRODUCING PYRROLE DERIVATIVE, AND INTERMEDIATE THEREOF
摘要 The present invention provides a method for producing an atropisomer of a pyrrole derivative having excellent mineralocorticoid receptor antagonistic activity, and an intermediate thereof. A method for producing an atropisomer of a pyrrole derivative using a compound represented by (B) [wherein R 1 represents a C1-C4 alkyl group, and R 2 represents a 2-hydroxyethyl group or a carboxymethyl group] as a production intermediate.
申请公布号 EP3040330(A1) 申请公布日期 2016.07.06
申请号 EP20140839943 申请日期 2014.08.26
申请人 DAIICHI SANKYO COMPANY, LIMITED 发明人 WATANABE, MASASHI;NAGASAWA, HIROSHI;SATO, NORITADA
分类号 C07D207/456;C07B57/00;C12P41/00 主分类号 C07D207/456
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