发明名称 |
AROMATIC COMPOUND |
摘要 |
Provided is a novel aromatic ring compound having a GPR40 agonist activity and a GLP-1 secretagogue action. A compound represented by the formula:
wherein each symbol is as described in the DESCRIPTION, or a salt thereof has a GPR40 agonist activity and a GLP-1 secretagogue action, is useful for the prophylaxis or treatment of cancer, obesity, diabetes, hypertension, hyperlipidemia, cardiac failure, diabetic complications, metabolic syndrome, sarcopenia and the like, and affords superior efficacy. |
申请公布号 |
EP3031799(A1) |
申请公布日期 |
2016.06.15 |
申请号 |
EP20140834225 |
申请日期 |
2014.08.08 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED |
发明人 |
AIDA, JUMPEI;YOSHITOMI, YAYOI;HITOMI, YUKO;NOGUCHI, NAOYOSHI;HIRATA, YASUHIRO;FURUKAWA, HIDEKI;SHIBUYA, AKITO;WATANABE, KOJI;MIYAMOTO, YASUFUMI;OKAWA, TOMOHIRO;TAKAKURA, NOBUYUKI;MIWATASHI, SEIJI |
分类号 |
C07D211/22;A61K31/451;A61K31/453;A61K31/4535;A61K31/454;A61K31/4545;A61K31/497;A61K31/506;A61K31/5377;A61P3/10;A61P43/00;C07D401/10;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D413/10;C07D413/14;C12N15/09 |
主分类号 |
C07D211/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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