| 发明名称 |
Tetrahydroquinoline compositions as BET bromodomain inhibitors |
| 摘要 |
The present invention relates to inhibitors of bromo and extra terminal (BET) bromodomains that are useful for the treatment of cancer, inflammatory diseases, diabetes, and obesity, having Formula (I): wherein W, X, Y, Z, R |
| 申请公布号 |
AU2014348191(A1) |
申请公布日期 |
2016.06.02 |
| 申请号 |
AU20140348191 |
申请日期 |
2014.11.18 |
| 申请人 |
FORMA THERAPEUTICS INC. |
发明人 |
BAIR, KENNETH W.;HERBERTZ, TORSTEN;KAUFFMAN, GOSS STRYKER;KAYSER-BRICKER, KATHERINE J.;LUKE, GEORGE P.;MARTIN, MATTHEW W.;MILLAN, DAVID S.;SCHILLER, SHAWN E. R.;TALBOT, ADAM C. |
| 分类号 |
C07D401/02;A61K31/47;A61K31/4709;C07D401/14 |
主分类号 |
C07D401/02 |
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