发明名称 SUBSTANTIALLY PURE VEMURAFENIB AND ITS SALTS
摘要 The present Invention relates to a process for the preparation substantially pure propane- 1 -sulfonicacid- { 3 -[5 -(4-chiorophenyI)-1 H-pyrrolo [2,3-b]pyridine-3 -carbonyl]-2,4-difluoro-phenyl} -amide or Vemurafenib of Formula (1), The present invention further relates to a process for the preparation substantially pure propane- 1 -sulfonic acid- { 3 - [5-(4-chlorophenyi)-1H-pyrrolo [2,3-b]pyridine-3 -carbonyl] -2,4-difluoro-phenyl} -amide trifluoro methane sulfonic acid salt or Vemurafenib triflate of Formula (VII).
申请公布号 WO2016083956(A1) 申请公布日期 2016.06.02
申请号 WO2015IB58964 申请日期 2015.11.19
申请人 SHILPA MEDICARE LIMITED 发明人 PUROHIT, PRASHANT;NAGNNATH, KOKARE;YENIREDDY, VEERA REDDY;AKSHAY KANT, CHATURVEDI
分类号 A61K31/437;C07D471/04 主分类号 A61K31/437
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