发明名称 PYRAZOLYL QUINAZOLINE KINASE INHIBITORS
摘要 The invention relates to new compounds, which are quinoxaline derivatives of formula Ito pharmaceutical compositions comprising said compounds, to processes for the preparation of said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
申请公布号 EA023222(B1) 申请公布日期 2016.05.31
申请号 EA20120091143 申请日期 2011.04.28
申请人 ASTEX THERAPEUTICS LIMITED 发明人 SAXTY GORDON;MURRAY CHRISTOPHER, WILLIAM;BERDINI VALERIO;BESONG GILBERT, EBAI;HAMLETT CHRISTOPHER, CHARLES, FREDERICK;JOHNSON CHRISTOPHER, NORBERT;WOODHEAD STEVEN, JOHN;READER MICHAEL;REES DAVID, CHARLES;MEVELLEC LAURENCE, ANNE;ANGIBAUD PATRICK, RENE;FREYNE EDDY, JEAN, EDGARD;GOVAERTS TOM, CORNELIS, HORTENSE;WEERTS JOHAN, ERWIN, EDMOND;PERERA TIMOTHY, PIETRO, SUREN;GILISSEN RONALDUS, ARNODUS, HENDRIKA, JOSEPH;WROBLOWSKI BERTHOLD;LACRAMPE JEAN, FERNAND, ARMAND;PAPANIKOS ALEXANDRA;QUEROLLE OLIVER, ALEXIS, GEORGES;PASQUIER ELISABETH, THERESE, JEANNE;PILATTE ISABELLE, NOELLE, CONSTANCE;BONNET PASCAL, GHISLAIN, ANDRE;EMBRECHTS WERNER, CONSTANT, JOHAN;AKKARI RHALID;MEERPOEL LIEVEN
分类号 C07D403/04;A61K31/498;A61P35/00;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D487/08 主分类号 C07D403/04
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