SOLID PHASE SYNTHESIS OF CYCLIC AMINO ACID MOLECULES
摘要
The present invention relates to cyclic amino acid molecules and methods of preparing the same, and in particular the macrocyclization of amino acids or linear peptides bound to a solid support.
申请公布号
WO2016079682(A1)
申请公布日期
2016.05.26
申请号
WO2015IB58903
申请日期
2015.11.17
申请人
ENCYCLE THERAPEUTICS;GOVERNING COUNCIL OF THE UNIVERSITY OF TORONTO;UNIVERSITE DE SHERBROOKE
发明人
HICKEY, JENNIFER L.;MANCUSO, JOHN;MARSAULT, ERIC;ROUGHTON, ANDREW L.;TREDER, ADAM P.;TREMBLEY, MARIE-CLAUDE J.;YUDIN, ANDREI K.;ZARETSKY, SERGE