发明名称 Process of producing cycloalkylcarboxamido-indole compounds
摘要 PROCESS OF PRODUCING CYCLOALKYLCARBOXAMIDO-INDOLE Abstract The present invention features processes for preparing compounds, such as (R)-1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-N-(1-(2,3-dihydroxypropyl)-6-fluoro-2 (1-hydroxy-2-methylpropan-2-yl)-1H-indol-5-yl)cyclopropanecarboxamide (Compound I), useful for treating CFTR mediated diseases such as cystic fibrosis.
申请公布号 AU2016202569(A1) 申请公布日期 2016.05.19
申请号 AU20160202569 申请日期 2016.04.22
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 LEE, ELAINE CHUNGMIN;TANOURY, GERALD J.;HARRISON, CRISTIAN;LITTLER, BENJAMIN JOSEPH;ROSE, PETER JAMISON;HUGHES, ROBERT MICHAEL;JUNG, YOUNG CHUN;SIESEL, DAVID ANDREW;BELMONT, DANIEL T.
分类号 C07D209/12;C07D317/60;C07D405/12 主分类号 C07D209/12
代理机构 代理人
主权项
地址