| 发明名称 |
HDAC INHIBITORS |
| 摘要 |
Compounds of formula (I) inhibit HDAC activity:;;wherein A, B and D independently represent ═C— or ═N—; W is a divalent radical —CH═CH— or CH2CH2—; R1 is an ester group; R2 is the side chain of a natural or non-natural alpha-amino acid; z is 0 or 1; and Y, L1, and X1 are as defined in the claims. |
| 申请公布号 |
US2016137594(A1) |
申请公布日期 |
2016.05.19 |
| 申请号 |
US201615004039 |
申请日期 |
2016.01.22 |
| 申请人 |
GlaxoSmithKline Intellectual Property Development Limited |
发明人 |
DAVIDSON Alan Hornsby;MOFFAT David Festus Charles;DAY Francesca Ann;DONALD Alastair David Graham |
| 分类号 |
C07C259/06;C07D241/04;C07D211/58;C07D211/34;C07C311/19;C07D213/56 |
主分类号 |
C07C259/06 |
| 代理机构 |
|
代理人 |
|
| 主权项 |
|
| 地址 |
Brentford GB |
