发明名称 |
Synthesis of trans-8-chloro-5-methyl-1 -[4-(Pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10b-tetraaza-benzo[e]azulene and crytalline forms thereof |
摘要 |
The present invention provides processes to manufacture substituted l-[4-(Pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10b- tetraaza-benzo[e]azulenes. Also disclosed are compounds useful as intermediates in the methods of the invention. |
申请公布号 |
AU2014359409(A1) |
申请公布日期 |
2016.05.19 |
申请号 |
AU20140359409 |
申请日期 |
2014.12.01 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
ROTHENHAEUSLER, BENNO;TRUSSARDI, RENE;HOFFMANN-EMERY, FABIENNE;SCHWITTER, URS;ADAM, JEAN-MICHEL;GRASSMANN, OLAF;HARTUNG, THOMAS;RAN, FREDERIC;DIODONE, RALPH;PFLEGER, CHRISTOPHE;BARTELS, BJOERN |
分类号 |
C07D487/04;A61K31/5517;A61P25/00 |
主分类号 |
C07D487/04 |
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