发明名称 Synthesis of trans-8-chloro-5-methyl-1 -[4-(Pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10b-tetraaza-benzo[e]azulene and crytalline forms thereof
摘要 The present invention provides processes to manufacture substituted l-[4-(Pyridin-2-yloxy)-cyclohexyl]-5,6-dihydro-4H-2,3,5,10b- tetraaza-benzo[e]azulenes. Also disclosed are compounds useful as intermediates in the methods of the invention.
申请公布号 AU2014359409(A1) 申请公布日期 2016.05.19
申请号 AU20140359409 申请日期 2014.12.01
申请人 F. HOFFMANN-LA ROCHE AG 发明人 ROTHENHAEUSLER, BENNO;TRUSSARDI, RENE;HOFFMANN-EMERY, FABIENNE;SCHWITTER, URS;ADAM, JEAN-MICHEL;GRASSMANN, OLAF;HARTUNG, THOMAS;RAN, FREDERIC;DIODONE, RALPH;PFLEGER, CHRISTOPHE;BARTELS, BJOERN
分类号 C07D487/04;A61K31/5517;A61P25/00 主分类号 C07D487/04
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