发明名称 TRICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS
摘要 The present invention relates to tricyclic heterocycles of Formula (I), which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer.
申请公布号 EP3019502(A1) 申请公布日期 2016.05.18
申请号 EP20140747194 申请日期 2014.07.07
申请人 INCYTE HOLDINGS CORPORATION 发明人 COMBS, ANDREW P.;YUE, EDDY W.;SPARKS, RICHARD B.;MADUSKUIE, JR., THOMAS P.
分类号 C07D498/06;A61K31/5383;A61P29/00;A61P31/00;A61P35/00 主分类号 C07D498/06
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