发明名称 |
TRICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS |
摘要 |
The present invention relates to tricyclic heterocycles of Formula (I), which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer. |
申请公布号 |
EP3019502(A1) |
申请公布日期 |
2016.05.18 |
申请号 |
EP20140747194 |
申请日期 |
2014.07.07 |
申请人 |
INCYTE HOLDINGS CORPORATION |
发明人 |
COMBS, ANDREW P.;YUE, EDDY W.;SPARKS, RICHARD B.;MADUSKUIE, JR., THOMAS P. |
分类号 |
C07D498/06;A61K31/5383;A61P29/00;A61P31/00;A61P35/00 |
主分类号 |
C07D498/06 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|